Aladinskiy Vladimir A.
Количество цитирований статей в журналах по данным
Web of Science: 62,
Scopus: 89
IstinaResearcherID (IRID): 21391630
Деятельность
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Статьи в журналах
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2020
Identification of pyrrolo-pyridine derivatives as novel class of antibacterials
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Veselov Mark S.,
Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Ayginin Andrey A.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Chemeris Alexey V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Maklakova Svetlana Yu,
Bezrukov Dmitry S.,
Filkov Gleb I.,
Zainullina Liana F.,
Maximova Marina A.,
Zileeva Zulfiya R.,
Kartsev Victor G.,
Vakhitova Yulia V.,
Dontsova Olga A.
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в журнале Molecular Diversity, издательство Springer Nature (Switzerland), том 24, № 1, с. 233-239
DOI
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2020
Synthesis and biological activity of 5-aryliden-2-thiohydantoin S-aryl derivatives
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Finko Alexander V.,
Skvortsov Dmitry A.,
Laikov Dimitri N.,
Averochkin Gleb M.,
Dlin Egor A.,
Kalinina Marina A.,
Aladinskiy Vladimir A.,
Vorobyeva Nataliya S.,
Mironov Andrei V.,
Beloglazkina Elena K.,
Zyk Nikolay V.,
Ivanenkov Yan A.,
Majouga Alexander G.
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в журнале Bioorganic Chemistry, издательство Academic Press (United States), том 100, с. 103900
DOI
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2019
2-Pyrazol-1-yl-thiazole derivatives as novel highly potent antibacterials
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Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Ayginin Andrey A.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Sadovnikov Sergey V.,
Rustam Matniyazov,
Sofronova Alina A.,
Malyshev Alexander S.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Dmitrii Lukianov,
Svetlana Iarovenko,
Bezrukov Dmitry S.,
Baymiev Andrey Kh,
Dontsova Olga A.
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в журнале Journal of Antibiotics, издательство Japan Antibiotics Research Association/Nihon Koseibusshitsu Gakujutsu Kyogikai (Japan), том 72, с. 827-833
DOI
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2019
Deep learning enables rapid identification of potent DDR1 kinase inhibitors
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Zhavoronkov Alex,
Ivanenkov Yan A.,
Aliper Alex,
Veselov Mark S.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasiya V.,
Terentiev Victor A.,
Polykovskiy Daniil A.,
Kuznetsov Maksim D.,
Asadulaev Arip,
Volkov Yury,
Zholus Artem,
Shayakhmetov Rim R.,
Zhebrak Alexander,
Minaeva Lidiya I.,
Zagribelnyy Bogdan A.,
Lee Lennart H.,
Soll Richard,
Madge David,
Xing Li,
Guo Tao,
Aspuru-Guzik Alán
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в журнале Nature Biotechnology, издательство Nature Publishing Group (United Kingdom)
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2019
Identification of N-Substituted Triazolo-azetidines as Novel Antibacterials using pDualrep2 HTS Platform
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Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Ayginin Andrey A.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Chemeris Alexey V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Malyshev Alexander S.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Bezrukov Dmitry S.,
Filkov Gleb I.,
Puchinina Maria M.,
Zainullina Liana F.,
Maximova Marina A.,
Zileeva Zulfiya R.,
Vakhitova Yulia V.,
Dontsova Olga A.
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в журнале Combinatorial Chemistry and High Throughput Screening, издательство Bentham Science Publishers (Netherlands), том 22, № 5, с. 346-354
DOI
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2019
Identification of Novel Antibacterials Using Machine Learning Techniques
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Ivanenkov Yan A.,
Zhavoronkov Alex,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Ayginin Andrey A.,
Kartsev Victor G.,
Skvortsov Dmitry A.,
Chemeris Alexey V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Malyshev Alexander S.,
Filkov Gleb I.,
Bezrukov Dmitry S.,
Zagribelnyy Bogdan A.,
Putin Evgeny O.,
Puchinina Maria M.,
Dontsova Olga A.
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в журнале Frontiers in pharmacology, издательство Frontiers Media] ([Lausanne, Switzerland), том 10, с. e913
DOI
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2019
Large-scale high-throughput screening revealed 5'-(carbonylamino)-2,3'-bithiophene-4'-carboxylate as novel template for antibacterial agents
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Ivanenkov YA,
Yamidanov RS,
Osterman IA,
Sergiev PV,
Aladinskiy VA,
Aladinskaya AV,
Terentiev VA,
Veselov MS,
Ayginin AA,
Skvortsov DA,
Komarova ES,
Zagribelnyy BA,
Baimiev AK,
Shvetc KY,
Sofronova AA,
Machulkin AE,
Petrov RA,
Zainullina LF,
Maximova MA,
Zileeva ZR,
Vakhitova YV,
Bezrukov DS,
Puchinina MM,
Dontsova OA
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в журнале Current Drug Discovery Technologies, издательство Bentham Science Publishers (Netherlands)
DOI
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2019
Substituted Furanocoumarins as Novel Class of Antibacterial Translation Inhibitors
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Ivanenkov Yan A.,
Yamidanov Renat S.,
Osterman Ilya A.,
Sergiev Petr V.,
Ayginin Andrey A.,
Aladinskiy Vladimir A.,
Aladinskaya Anastasia V.,
Terentiev Victor A.,
Veselov Mark S.,
Skvortsov Dmitry A.,
Komarova Katerina S.,
Chemeris Alexey V.,
Zainullina Liana F.,
Maximova Marina A.,
Zileeva Zulfiya R.,
Vakhitova Yulia V.,
Baimiev Alexey Kh,
Sofronova Alina A.,
Machulkin Alexey E.,
Petrov Rostislav A.,
Bezrukov Dmitry S.,
Puchinina Maria M.,
Dmitrii Lukianov A.,
Dontsova Olga A.
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в журнале Combinatorial Chemistry and High Throughput Screening, издательство Bentham Science Publishers (Netherlands), том 22, № 6, с. 400-410
DOI
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2018
Entangled Conditional Adversarial Autoencoder for de-Novo Drug Discovery
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Polykovskiy Daniil,
Zhebrak Alexander,
Vetrov Dmitry,
ivanenkov yan,
Aladinskiy Vladimir,
Bozdaganyan Marine,
Mamoshina Polina,
Aliper Alex,
Zhavoronkov Alex,
Kadurin Artur
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в журнале Molecular Pharmaceutics, издательство American Chemical Society (United States)
DOI
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2016
Small-molecule PSMA ligands. Current state, SAR and perspectives
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Machulkin Alexey E.,
Ivanenkov Yan A.,
Aladinskaya Anastasia V.,
Veselov Mark S.,
Aladinskiy Vladimir A.,
Beloglazkina Elena K.,
Koteliansky Victor E.,
Shakhbazyan Artem G.,
Sandulenko Yuri B.,
Majouga Alexander G.
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в журнале Journal of Drug Targeting, издательство Taylor & Francis (United Kingdom), том 24, № 8, с. 679-693
DOI
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Доклады на конференциях